Term
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Definition
| Direct cholinergic agonist (M+N). Ultra short acting via IV. |
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Term
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Definition
| Direct muscarinic Ach antagonist. short acting, renal excretion. M1-M5. widely distributed, incl CNS. Oral, parenteral, and opthalmic. Side effects are dose dependent. small dose decreses HR, larger dose increases HR. decreased sweating, pupillary dilation, dry mouth, tachycardia, enhanced AV node conduction, bronchodilation, decused sweating (hyperthermia in kids), reduced salivation, sedation and reduces parkinsons rigidity (CNS). Uses: acute treatment of bradycardia and AV block. Also, use to treat organophosphate poisining. Used to be used to treat asthma and allergies. |
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Term
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Definition
| direct muscarinic Ach inhibitor. oral. Use: parkinsons disease. |
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Term
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Definition
| Direct cholinergic agonist (M). Oral, longer acting than Ach. Use: postoperative gastic atony and non obstructive urinary retention, |
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Term
| Carbamylcholine = carbachol |
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Definition
| Direct cholinergic agonist (M+N). |
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Term
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Definition
| ACE inhibitor. 4* amide. reversible. short acting minutes, parenteral. Use: diagnostic for Myesthenia gravis. |
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Term
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Definition
| indirect muscarinic Ach antagonist. ganglionic blocer. old treatment for HTN, side effects of combined S and PS effects. |
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Term
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Definition
| direct muscarinic Ach inhibitor. 4* amine, inhaled aerosol. Uses: asthma, COPD. |
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Term
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Definition
| ACE inhibitor. irreversible. Organophosphate. long acting, lipid soluble. |
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Term
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Definition
| Indirect muscarinic receptor antagonist. ganglionic blocker. previously used to treat HTN, but causes symptoms of both S and PS. |
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Term
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Definition
| non-selective muscarinic receptor agonist |
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Term
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Definition
| ACE inhibitor. reversible. Carbamate Ester. mins-hrs, oral and parenteral. Use: treatment for myesthenia gravis. Also, paralytic iileus and atonic bladder. |
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Term
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Definition
| Nicotine agonist, cigurretes. |
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Term
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Definition
| direct muscarinic Ach inhibitor. oral and transdermal. uses: overactive urinary bladder and spastic bladder of paraplegic. |
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Term
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Definition
| nicotinic Ach receptor blocker. Use: surgery and ECt. |
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Term
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Definition
| ACE inhibitor, irreversible. Organophosphate. long acting. lipid soluble. toxins! |
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Term
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Definition
| ACE inhibitor, reversible. Carbamate Ester. mins-hrs, parenteral. Use: treat anticholinergic poisining. CNS effects (vs pyridostigmine). |
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Term
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Definition
| Direct cholinergic agonist (M). Opthalmic or oral. Use: chronic glaucoma. |
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Term
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Definition
| can hydrolyze organophosphate-ACE bond, used to treat nerve gas if given soon enough. |
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Term
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Definition
| ACE inhibitor, reversible. Carbamate ester. hours. oral and parenteral. Use: treatment for myesthenia gravis and prophylaxis for organophosphate poisining. No CNS effects. |
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Term
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Definition
| direct muscarinic ACh antagonist. oral, parenteral, opthalmmic, and transdermal. Use: motion sickness. |
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Term
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Definition
| nicotinic Ach receptor blocker. Use: surgery and ECT |
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Term
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Definition
| Indirec antag, ganglionic blocker |
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Term
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Definition
| direct muscarinic Ach inhibitor. opthalmic. Short acting, so use for pupillary dilation. careful, can precipitate glaucoma in pre-disposed ppl. |
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Term
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Definition
| nerve gas. Organophosphate, ACE inhibitor. |
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