Term
|
Definition
| Carbamazepine (autoinducer), Rifampin, Phenytoin, Phenobarbita,l St. Johns Wort |
|
|
Term
|
Definition
| Amiodarone Cimetidine Clarithromycin Erythromycin Grapefruit Juice Itraconazole Ketoconazole |
|
|
Term
|
Definition
| Carbamazepine Glucocorticoids Phenytoin Rifampin Ritonavir |
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|
Term
|
Definition
| Cimetidine Ciprofloxacin Clarithromycin Enoxacin Erythromycin Fluvoxamine Ofloxacine Ticlopidine |
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|
Term
|
Definition
| Hydrocarbons (cigarette smoke) |
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Term
|
Definition
| Clozapine Cyclobenzaprine Fluvoxamine Imipramine Mexiletine Propranolol Theophylline |
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|
Term
| Most important substrate of 1A2 |
|
Definition
|
|
Term
| 1A2 mostly metabolizes what medication types? |
|
Definition
|
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Term
|
Definition
| Diclofenac Ibuprofen Losartan Naproxen Phenytoin Piroxicam Sulfamethoxazole Warfarin |
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|
Term
|
Definition
|
|
Term
|
Definition
| Amiodarone Fluconazole Fluoxetine(SSRI) Isoniazid (TB) Paroxetine (SSRI) Ticlopidine (SSRI) Zafirlukast |
|
|
Term
| Two most important inhibitors of 2C9 |
|
Definition
| Amiodarone and flucanazole |
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|
Term
|
Definition
|
|
Term
|
Definition
| Amitriptyline Clomipramine Ciclophosphamide Diazepam Imiprimine Lansoprazole Omeprazole Phenytoin Clopidogrel |
|
|
Term
| Most important substrate of 2C19 |
|
Definition
|
|
Term
|
Definition
| Carbamazepine Norethindrone |
|
|
Term
|
Definition
| Cimetidine Fluoxetine Fluvoxamine Ketoconazole Lansoprazole Omeprazole Paroxetine Ticlopidine |
|
|
Term
| 2C19 is inhibited by what classes? |
|
Definition
| SSRIs (paraxetine) and PPIs |
|
|
Term
|
Definition
| APAP Chlorzoxazone Ethanol Enflurane Halothane Isolurane |
|
|
Term
|
Definition
| Isonizid and Chronic Ethanol |
|
|
Term
|
Definition
| Amiodarone Fluoxetine Haloperidol Indinavir Paroxetine Quinidine Ritonavir Sertraline |
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Term
|
Definition
|
|