Term
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Definition
| Anxiolytic, Rarely Used anymore |
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Term
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Definition
| Ultra-Short-Acting Barb, used in Induction of Anesthesia |
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Term
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Definition
| Short-Acting Barb, Anxiolytic, Metabolism and Renal Excretion are Major Paths to terminate Drug Action |
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Term
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Definition
| Depress Medullary Respiratory Center, Potentiated by Alcohol, Induces Enzymes altering self/non-self drug metabolism, Tolerance, Dependence (Severe Withdrawal) |
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Term
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Definition
| Long T 1/2, Causes Skeletal Muscle Relaxation |
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Term
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Definition
| Benzodiazepine with Intermediate Elimination (T 1/2) |
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Term
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Definition
| Benzodiazepine with Intermediate Elimination (T 1/2) Does NOT require Phase 1 Metabolism therefore is safer in patients with hepatic failure |
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Term
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Definition
| Benzo used to treat Panic Attacks |
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Term
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Definition
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Term
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Definition
| Don't Cause Anesthesia, Less Severe Withdrawal, Can Cause both CNS Depression or paradoxical CNS Activation and nightmares, Tolerance and Dependance, Selflimited Action |
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Term
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Definition
| @ high doses can directly activate Cl channels |
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Term
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Definition
| Benzodiazepine Receptor Antagonist |
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Term
| Desmethydiazepam and Nordazepam |
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Definition
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Term
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Definition
| Slow Onset Anxiolytic with low addiction potential, Does not potentiate alcohol CNS Depression, Minimal Sedation, Stimulates 5-HT1a receptor (No action on GABA) |
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Term
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Definition
| Hypnotic that Works @ Benzodiazepine Receptor, No rebound insomnia, No Withdrawal, Minimal Tolerance may occur |
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Term
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Definition
| Mirrors Benzo Action by binding GABA Receptors at the same site BUT no tolerance for at least 6 months making this hypnotic useful for treating Chronic Insomnia |
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